• Title of article

    Amine-catalyzed direct asymmetric Mannich-type reactions

  • Author/Authors

    Notz، نويسنده , , Wolfgang and Sakthivel، نويسنده , , Kandasamy and Bui، نويسنده , , Tommy and Zhong، نويسنده , , Guofu and Barbas III، نويسنده , , Carlos F، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2001
  • Pages
    3
  • From page
    199
  • To page
    201
  • Abstract
    Three chiral cyclic secondary amines are shown to be catalysts for the direct asymmetric Mannich-type reaction of acetone with a variety of preformed aldimines derived from o-anisidine. A simple one-pot three-component reaction procedure consisting of aldehyde, acetone, p-anisidine and an amine catalyst provides the corresponding β-amino ketones with 50–89% ee under very mild conditions.
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2001
  • Journal title
    Tetrahedron Letters
  • Record number

    1641010