• Title of article

    Michael addition of amines to vinyl sulfonamides on solid support

  • Author/Authors

    Makara، نويسنده , , Gergely M and Ma، نويسنده , , Yao، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2001
  • Pages
    3
  • From page
    4123
  • To page
    4125
  • Abstract
    A solid phase synthesis for Michael addition of amines to vinylsulfonamides has been developed. The method enables synthesis of β-aminosulfonamides with high yields and purity. Further functionalization of adducts derived from primary amines is demonstrated.
  • Keywords
    combinatorial , sulfonamides , Michael addition , solid phase
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2001
  • Journal title
    Tetrahedron Letters
  • Record number

    1645293