• Title of article

    Diastereocontrolled reduction of cyclic β-enaminones. A new diastereoselective route to 2,6-disubstituted piperidines

  • Author/Authors

    Fréville، نويسنده , , Stéphanie and Delbecq، نويسنده , , Philippe and Thuy، نويسنده , , Vu Moc and Petit، نويسنده , , Huguette and Célérier، نويسنده , , Jean Pierre and Lhommet، نويسنده , , Gérard، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2001
  • Pages
    3
  • From page
    4609
  • To page
    4611
  • Abstract
    A new diastereoselective synthesis of 2,6-disubstituted piperidinic alkaloids is presented. Three natural compounds, the (−)-pinidinone 1a, the (+)-dihydropinidine 1b and the (−)-pinidinol 1c were prepared from optically pure (6R)-6-methylpiperidin-2-one 2. This method is based on the chemo- and diastereocontrolled reductions of an exocyclic β-enamino ketone.
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2001
  • Journal title
    Tetrahedron Letters
  • Record number

    1645687