Author/Authors :
Caballero، نويسنده , , Esther and Longieras، نويسنده , , Nicolas and Zausa، نويسنده , , Elodie and del Rey، نويسنده , , Benedicto and Medarde، نويسنده , , Manuel and Tomé، نويسنده , , Fernando، نويسنده ,
Abstract :
The preparation of (E)-1-(3-indolyl)-3-tert-butyldimethylsiloxy-1,3-butadienes and their Diels–Alder reaction with selected dienophiles at room temperature is described. The utility of these heteroaryldienes for the construction of different (3-indolyl)-planar systems is shown by the synthesis of a grooved analogue of arcyriaflavin A.
Keywords :
Dienes , Diels–Alder reactions , indoles , Alkaloids
