Title of article
A new reagent and its polymer-supported variant for the amidination of amines
Author/Authors
Drنger، نويسنده , , Gerald and Solodenko، نويسنده , , Wladimir and Messinger، نويسنده , , Josef and Schِn، نويسنده , , Uwe and Kirschning، نويسنده , , Andreas، نويسنده ,
Issue Information
هفته نامه با شماره پیاپی سال 2002
Pages
3
From page
1401
To page
1403
Abstract
New reagents for the high yielding amidination of primary and secondary amines are described. By attaching a benzyl substituent to the 3,5-dimethyl-1H-pyrazole-1-carboxamidine ring, a reagent 1 is obtained which allows easy work-up after amidination because of solubility of byproducts in organic solvents. In addition, the polystyrene-bound analogue 2 was prepared which allows amidination of various amines with high purity.
Journal title
Tetrahedron Letters
Serial Year
2002
Journal title
Tetrahedron Letters
Record number
1650012
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