• Title of article

    Synthesis of a new chelating agent derived from phenylenediamine for application in radioimmunotherapy

  • Author/Authors

    Gouin، نويسنده , , Sébastien G. and Gestin، نويسنده , , Jean-François and Reliquet، نويسنده , , Alain and Meslin، نويسنده , , Jean Claude and Deniaud، نويسنده , , David، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2002
  • Pages
    3
  • From page
    3003
  • To page
    3005
  • Abstract
    We report the synthesis of a new diethylenetriaminepentaacetic acid (DTPA) analogue, Ph-DTPA, possessing an aromatic rigid skeleton. This precursor of a bifunctional chelating agent was synthesized by elaboration of the intermediate N-(o-aminophenyl)ethylenediamine and obtained in five steps with an overall yield of 42%. Preliminary complexation studies between Ph-DTPA and 153Sm has been carried out.
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2002
  • Journal title
    Tetrahedron Letters
  • Record number

    1651201