Title of article
Synthesis of C-glycosyl β-amino acids by asymmetric Mannich-type three-component reactions
Author/Authors
Dondoni، نويسنده , , Alessandro and Massi، نويسنده , , Alessandro and Sabbatini، نويسنده , , Simona and Bertolasi، نويسنده , , Valerio، نويسنده ,
Issue Information
هفته نامه با شماره پیاپی سال 2004
Pages
4
From page
2381
To page
2384
Abstract
C-Galactosyl and C-ribosyl β-amino acids were prepared by one-pot InCl3-catalyzed Mannich-type three-component condensation (3CC) by combining the corresponding formyl C-glycoside, p-methoxybenzyl amine, and a ketene silyl acetal. In each case the reaction was highly stereoselective and afforded only one single product in good to excellent yields.
Keywords
multicomponent reaction , Mannich reaction , Unnatural peptides , C-Glycosyl ?-amino acids
Journal title
Tetrahedron Letters
Serial Year
2004
Journal title
Tetrahedron Letters
Record number
1657574
Link To Document