Author/Authors :
Li، نويسنده , , Jiayin and Liang، نويسنده , , Jiang-Lin and Chan، نويسنده , , Philip Wai Hong and Che، نويسنده , , Chi-Ming، نويسنده ,
Abstract :
Aziridination of a variety of alkenes with N-substituted hydrazines mediated by iodobenzene diacetate under mild conditions (K2CO3, CH2Cl2) and ambient temperature were achieved in good to excellent yields (up to 99%), and conversions. The practicality and simplicity of this C–N bond formation protocol was exemplified by its application to the aziridination of cholesteryl acetate in a stereoselective manner.
