Title of article
Preparation of 2-hydroxybenzamidines from 3-aminobenzisoxazoles
Author/Authors
Lepore، نويسنده , , Salvatore D and Schacht، نويسنده , , Aaron L and Wiley، نويسنده , , Michael R، نويسنده ,
Issue Information
هفته نامه با شماره پیاپی سال 2002
Pages
3
From page
8777
To page
8779
Abstract
2-Hydroxybenzamidines have been prepared from 3-aminobenzisoxazoles by reductive cleavage of the nitrogen–oxygen bond using catalytic hydrogenation, Zn/AcOH or NiCl2/NaBH4. This ring-opening reaction can be accomplished chemoselectively in the presence of a variety of hydrogenation-sensitive functional groups including an aryl bromide, benzyl carbamate, and olefin.
Journal title
Tetrahedron Letters
Serial Year
2002
Journal title
Tetrahedron Letters
Record number
1659265
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