Title of article
A facile synthesis of 4- and 6-chloromethyl-1H-indole-2-carboxylates: replacement of a sulfonic acid functionality by chlorine
Author/Authors
Pete، نويسنده , , Béla and Parlagh، نويسنده , , Gyula، نويسنده ,
Issue Information
هفته نامه با شماره پیاپی سال 2003
Pages
3
From page
2537
To page
2539
Abstract
Valuable new synthetic intermediates, 4- or 6-chloromethyl-1H-indole-2-carboxylates, were prepared by the elimination of SO2 from 2-ethoxycarbonyl-1H-indole-4- or 6-methanesulfonic acids, respectively, which are easily accessible by Fischer-type indolization.
Keywords
Fischer synthesis , 4-(chloromethyl)indoles , 6-(chloromethyl)indoles , Desulfination
Journal title
Tetrahedron Letters
Serial Year
2003
Journal title
Tetrahedron Letters
Record number
1661320
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