• Title of article

    Towards the synthesis of osteoclast inhibitor SB-242784

  • Author/Authors

    Conde، نويسنده , , Jose J. and McGuire، نويسنده , , Michael and Wallace، نويسنده , , Michael، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2003
  • Pages
    4
  • From page
    3081
  • To page
    3084
  • Abstract
    Osteoclast inhibitor SB-242784 (1) was prepared from pivotal indol intermediate 4. A ‘Stille’ cross coupling of organotin 2c with bromo acrylate 11 afforded diene 12 which was also obtained via a reduction–isomerization process of enyne 16. Bromoamide 3 was prepared from the corresponding acid 7 which was readily obtained from bromopyruvic acid.
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2003
  • Journal title
    Tetrahedron Letters
  • Record number

    1661646