• Title of article

    Electronic effect on the regioselectivity in the ring opening of para-substituted phenyloxiranes by acetylides

  • Author/Authors

    Shindo، نويسنده , , Mitsuru and Sugioka، نويسنده , , Tomoyuki and Shishido، نويسنده , , Kozo، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2004
  • Pages
    4
  • From page
    9265
  • To page
    9268
  • Abstract
    The electronic effect on the regioselectivity in the alkynylation of phenyloxiranes was investigated using three kinds of metal acetylides. BF3 mediated lithium acetylide provided either the α- or β-alkynylated products by controlling the effect of the para-substituents of the phenyloxiranes. LiClO4 mediated lithium acetylide and titanium acetylide, on the other hand, afforded predominantly the β- and α-products, respectively.
  • Keywords
    Lewis acid , Electronic effect , Oxirane , Alkynylation , regioselectivity
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2004
  • Journal title
    Tetrahedron Letters
  • Record number

    1844150