Title of article :
A practical entry to C18-constrained-E-ring analogues of methyllycaconitine (MLA): a concise new stereoselective approach to 8-oxa-decahydroisoquinolines accompanied by a simple microwaves-assisted synthesis of the succinimidobenzoate appendage of MLA
Author/Authors :
Simoni، نويسنده , , Daniele and Rossi، نويسنده , , Marcello and Rondanin، نويسنده , , Riccardo and Baruchello، نويسنده , , Riccardo and Grisolia، نويسنده , , Giuseppina and Eleopra، نويسنده , , Marco and Giovannini، نويسنده , , Riccardo and Bozzoli، نويسنده , , Andrea and Davalli، نويسنده , , Silvia and Di Fabio، نويسنده , , Romano and Donati، نويسنده , , Daniele، نويسنده ,
Issue Information :
هفته نامه با شماره پیاپی سال 2005
Pages :
4
From page :
759
To page :
762
Abstract :
A Mannich-type intramolecular cyclization afforded access to a 8-oxa-decahydroisoquinoline heterocyclic system. Good stereoselectivity was observed. A promising microwave-assisted synthesis of the methylsuccinimidobenzoate moiety of methyllycaconitine has also been carried out.
Keywords :
Methyllycaconitine , Nicotinic acetylcholine receptor antagonists , microwave-assisted chemistry , Decahydroisoquinoline synthesis
Journal title :
Tetrahedron Letters
Serial Year :
2005
Journal title :
Tetrahedron Letters
Record number :
1844612
Link To Document :
https://search.isc.ac/dl/search/defaultta.aspx?DTC=10&DC=1844612
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