• Title of article

    Selective bifunctionalization of pyrido[2,3-d]pyrimidines in positions 2 and 4 by SNAr and palladium-catalyzed coupling reactions

  • Author/Authors

    Lavecchia، نويسنده , , G. and Berteina-Raboin، نويسنده , , S. and Guillaumet، نويسنده , , G.، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2005
  • Pages
    5
  • From page
    5851
  • To page
    5855
  • Abstract
    Selective disubstitution of 2,4-dichloropyrido[2,3-d]pyrimidine with various nucleophiles was investigated. Suzuki and Stille cross-coupling reactions on monosubstituted compound 4-tert-butylamino-2-chloro-pyrido[2,3-d]pyrimidine were performed in high yields.
  • Keywords
    Suzuki reaction , cross-coupling , Stille reaction , PALLADIUM , 3-d]pyrimidine , SNAr
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2005
  • Journal title
    Tetrahedron Letters
  • Record number

    1846510