• Title of article

    Diastereoselective synthesis of (2S∗)-2-[(R∗)-1H-indol-3-yl(phenyl)methyl]-2,3-dihydro-1H-inden-1-one

  • Author/Authors

    Semenov، نويسنده , , Boris B. and Novikov، نويسنده , , Kirill A. and Lysenko، نويسنده , , Konstantin A. and Kachala، نويسنده , , Vadim V.، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2006
  • Pages
    5
  • From page
    3479
  • To page
    3483
  • Abstract
    Double asymmetric induction in Michael reactions has been studied. Enantioselective alkylation of a cyclic ketone (1-indanone) with α-phenyl-nor-gramine was carried out. The relative configuration of (2S∗)-2-[(R∗)-1H-indol-3-yl(phenyl)methyl]-2,3-dihydro-1H-inden-1-one was established by X-ray diffraction. The relative configuration of (R∗,R∗,S∗)- and (S∗,R∗,S∗)-2-1H-indol-3-yl(phenyl)methyl]-2,3-dihydro-1H-inden-1-ols was established by 1H NMR studies.
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2006
  • Journal title
    Tetrahedron Letters
  • Record number

    1850338