• Title of article

    A new approach for the construction of a highly congested bicyclic system in polycyclic polyprenylated acylphloroglucinols (PPAPs)

  • Author/Authors

    Shimizu، نويسنده , , Yohei and Kuramochi، نويسنده , , Akiyoshi and Usuda، نويسنده , , Hiroyuki and Kanai، نويسنده , , Motomu and Shibasaki، نويسنده , , Masakatsu، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2007
  • Pages
    5
  • From page
    4173
  • To page
    4177
  • Abstract
    A highly congested bicyclo[3.3.1]nonanone core of polycyclic polyprenylated acylphloroglucinols was constructed using a stereoselective Claisen rearrangement and an intramolecular aldol reaction as the key steps. The stereochemistry of C-4 appeared to control the ground state conformation of the cyclohexenone core, which determined the diastereoselectivity in the Claisen rearrangement.
  • Keywords
    garsubellin A , Polycyclic polyprenylated acylphloroglucinols (PPAPs) , Claisen rearrangement , intramolecular aldol reaction , hyperforin
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2007
  • Journal title
    Tetrahedron Letters
  • Record number

    1855182