• Title of article

    Copper-catalyzed one-pot N-alkenylation and N-alkylation of amides: an efficient synthesis of substituted 2,3-dihydropyrroles

  • Author/Authors

    Zhou، نويسنده , , Xiaobo and Zhang، نويسنده , , Huimin and Yuan، نويسنده , , Jiwei and Mai، نويسنده , , Lugen and Li، نويسنده , , Yanzhong، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2007
  • Pages
    4
  • From page
    7236
  • To page
    7239
  • Abstract
    A novel copper-catalyzed synthesis of substituted 2,3-dihydropyrroles via one-pot N-alkenylation and N-alkylation of amides with 1,4-diiodobut-1-ene derivatives has been developed. The reactions proceed in good to high yields using CuI as the catalyst, K2CO3 as the base, and rac-trans-N,N′-dimethylcyclohexane-1,2-diamine as the ligand.
  • Keywords
    copper catalyst , N-Alkenylation , N-Alkylation , Amides , dihydropyrroles
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2007
  • Journal title
    Tetrahedron Letters
  • Record number

    1856765