Title of article
Synthesis of 1,1-disubstituted tetrahydro-β-carbolines from 2-methyleneaziridines
Author/Authors
Mumford، نويسنده , , Peter M. and Shiers، نويسنده , , Jason J. and Tarver، نويسنده , , Gary J. and Hayes، نويسنده , , Jerome F. and Shipman، نويسنده , , Michael، نويسنده ,
Issue Information
هفته نامه با شماره پیاپی سال 2008
Pages
3
From page
3489
To page
3491
Abstract
Ring opening of indole functionalised methyleneaziridines (3a–c, 7) with alcohols in the presence of boron trifluoride etherate leads to the formation of 1,1-disubstituted tetrahydro-β-carbolines in moderate to good yields (37–83%).
Keywords
Ring opening , Nitrogen Heterocycles , strained compounds , Pictet–Spengler , Aziridines
Journal title
Tetrahedron Letters
Serial Year
2008
Journal title
Tetrahedron Letters
Record number
1859337
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