• Title of article

    Organocatalytic asymmetric nitrocyclopropanation of α,β-unsaturated aldehydes

  • Author/Authors

    Vesely، نويسنده , , Jan and Zhao، نويسنده , , Gui-Ling and Bartoszewicz، نويسنده , , Agnieszka and Cَrdova، نويسنده , , Armando، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2008
  • Pages
    4
  • From page
    4209
  • To page
    4212
  • Abstract
    A novel organocatalytic highly enantioselective nitrocyclopropanation reaction of α,β-unsaturated aldehydes is presented. The 1-nitro-2-formylcyclopropane derivatives synthesized from this catalytic transformation were converted to the corresponding β-nitromethyl-acid esters, which are excellent precursors of GABA analogues such as Baclofen, by subsequent organocatalytic chemoselective ring-opening.
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2008
  • Journal title
    Tetrahedron Letters
  • Record number

    1859666