Author/Authors :
Wang، نويسنده , , Junke and Peng، نويسنده , , Feng and Jiang، نويسنده , , Ju-li and Lu، نويسنده , , Zhijin and Wang، نويسنده , , Le-yong and Bai، نويسنده , , Junfeng and Pan، نويسنده , , Yi، نويسنده ,
Abstract :
Employing N-(4,5-dihydrooxazol-2-yl)benzamide as novel and efficient ligand, the copper-catalyzed intramolecular cyclization of various substituted 1-acyl-3-(2-bromophenyl)thioureas could be successfully carried out under mild conditions. A variety of N-benzothiazol-2-yl-amides were synthesized in good to excellent yields.
Keywords :
Intramolecular cyclization , Copper , Thiourea , Benzothiazol-2-yl-amide