• Title of article

    Phenyl esters, preferred reagents for mono-acylation of polyamines in the presence of water

  • Author/Authors

    Pappas، نويسنده , , Kyrie and Zhang، نويسنده , , Xiang and Tang، نويسنده , , Wei and Fang، نويسنده , , Shiyue، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2009
  • Pages
    3
  • From page
    5741
  • To page
    5743
  • Abstract
    In the presence of water, several diamines and one triamine were mono-acylated at ambient to moderate temperatures using phenyl esters and a phenyl carbonate as acylation agents in good to excellent isolated yields. Both linear and cyclic polyamines were suitable substrates, and the acylating agents can be aryl and alkyl carboxylic acid esters.
  • Keywords
    water , Phenyl ester , Mono-acylation , Diamine , Piperazine
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2009
  • Journal title
    Tetrahedron Letters
  • Record number

    1866106