Author/Authors :
Laliberté، نويسنده , , Sébastien and Dornan، نويسنده , , Peter K. and Chen، نويسنده , , Austin، نويسنده ,
Abstract :
The synthesis of pyrazino[1,2-a]indoles via a palladium-catalyzed double allylic alkylation of indole-2-hydroxamates is described. The reaction conditions are very mild and allow for a wide variety of substitutions on the indole core.