• Title of article

    Asymmetric synthesis of (+)-chloriolide

  • Author/Authors

    Das، نويسنده , , Tapas and Jana، نويسنده , , Nandan and Nanda، نويسنده , , Samik، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2010
  • Pages
    4
  • From page
    2644
  • To page
    2647
  • Abstract
    An asymmetric synthesis of 12-membered ring macrolide, chloriolide has been accomplished by adopting a linear strategy. Lipase-catalyzed enzymatic kinetic resolution (EKR), asymmetric alkynylation using Trost pro-phenol catalyst followed by Yamaguchi macrolactonization has been successfully employed to achieve the target molecule.
  • Keywords
    Asymmetric alkynylation , Asymmetric total synthesis , macrolactonization , Medium ring macrolides , Enzymatic kinetic resolution (EKR)
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2010
  • Journal title
    Tetrahedron Letters
  • Record number

    1872157