Title of article
Synthesis of azepino[3,4b]indoles via the Plancher rearrangement
Author/Authors
Eisenbeis، نويسنده , , Shane A. and Phillips، نويسنده , , James R. and Rescek، نويسنده , , Diane and Oyola-Cintron، نويسنده , , Yatsandra and Kock، نويسنده ,
Issue Information
هفته نامه با شماره پیاپی سال 2010
Pages
3
From page
4303
To page
4305
Abstract
The reaction of benzyl 3-formylpiperidine-1-carboxylate and aryl hydrazines under standard Fisher Indole conditions followed by reductive work-up affords azepino[3,4b]indoles in moderate to good yields. The products are proposed to be derived via a Plancher rearrangement [(a) Plancher, G. Gazz. Chim. Ital. 1898, 28, II, 374; (b) Plancher, G. Atti. Accad. Lincei 1900, 9, 5, 115; (c) Boyd-Barrett, H. S. J. Chem. Soc. 1932, 321].
Keywords
Fisher indole , Plancher rearrangement , 4b]indoles
Journal title
Tetrahedron Letters
Serial Year
2010
Journal title
Tetrahedron Letters
Record number
1874016
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