Title of article
Direct C2-trifluoromethylation of indole derivatives catalyzed by copper acetate
Author/Authors
Shimizu، نويسنده , , Ryo and Egami، نويسنده , , Hiromichi and Nagi، نويسنده , , Tatsuya and Chae، نويسنده , , Jungha and Hamashima، نويسنده , , Yoshitaka and Sodeoka، نويسنده , , Mikiko، نويسنده ,
Issue Information
هفته نامه با شماره پیاپی سال 2010
Pages
3
From page
5947
To page
5949
Abstract
Direct C2-selective trifluoromethylation of indole derivatives was achieved with Togni’s hypervalent iodine reagent and CuOAc as a catalyst in MeOH under mild conditions, affording the desired C2-trifluoromethylated indoles in good yield (up to 90%).
Keywords
trifluoromethylation , indole , Catalysis , regioselective
Journal title
Tetrahedron Letters
Serial Year
2010
Journal title
Tetrahedron Letters
Record number
1875418
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