• Title of article

    Synthesis of 2,3-dihydro-1,4-dithiinyl nucleosides via Pummerer-type glycosidation

  • Author/Authors

    Paolella، نويسنده , , Concetta and D’Alonzo، نويسنده , , Daniele and Guaragna، نويسنده , , Annalisa and Cermola، نويسنده , , Flavio and Palumbo، نويسنده , , Giovanni، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2010
  • Pages
    4
  • From page
    6060
  • To page
    6063
  • Abstract
    A straightforward procedure for the preparation of nucleoside analogue 1 and its regioisomer 2 containing a dihydro-1,4-dithiin as sugar moiety has been accomplished in four steps by our readily available heterocyclic system 5. Nucleobase insertion was carried out by direct addition of N4-acetylcytosine to sulfoxide derivatives via Pummerer-type glycosidation reaction.
  • Keywords
    Heterocyclic nucleosides , Dithiins , Nucleoside analogues , Pummerer-type glycosidation
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2010
  • Journal title
    Tetrahedron Letters
  • Record number

    1875512