• Title of article

    Direct glycosylation with anomeric hydroxy sugars by activation with 3-fluorophthalic anhydride and trifluoromethanesulfonic anhydride

  • Author/Authors

    Baek، نويسنده , , Ju Yuel and Lee، نويسنده , , Bo-Young and Pal، نويسنده , , Rita and Lee، نويسنده , , Won-Yong and Kim، نويسنده , , Kwan Soo، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2010
  • Pages
    5
  • From page
    6250
  • To page
    6254
  • Abstract
    An efficient and direct one-pot glycosylation method using anomeric hydroxy sugars as glycosyl donors, employing 3-fluorophthalic anhydride and triflic anhydride as activating agents, has been developed. The present glycosylation utilizing 3-fluorophthalic anhydride resulted in few to no undesired self-condensed esters than the glycosylation using phthalic anhydride. Intermediates in the present glycosylation were identified by an NMR study.
  • Keywords
    glycosylation , Glycosyl fluorophthalate , 3-Fluorophthalic anhydride
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2010
  • Journal title
    Tetrahedron Letters
  • Record number

    1875663