• Title of article

    Synthesis of estradiol backbone mimics via the Stille reaction using copper(II) oxide as co-reagent

  • Author/Authors

    Flِistrup، نويسنده , , Erik and Goede، نويسنده , , Patrick and Strِmberg، نويسنده , , Roger and Malm، نويسنده , , Johan، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2011
  • Pages
    3
  • From page
    209
  • To page
    211
  • Abstract
    Sterically hindered biaryls and 2-phenylbenzo[b]thiophenes that can serve as templates for mimics of the estradiol backbone were prepared in modest to good yields by the Stille reaction using CuO as a co-reagent. Due to the neutral conditions applied in the Stille reaction, protection strategies were unnecessary for hydroxy containing coupling partners. Ligandless coupling conditions were also evaluated.
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2011
  • Journal title
    Tetrahedron Letters
  • Record number

    1876368