Title of article :
A concise synthesis of HIV integrase inhibitors bearing the dipyridone acid motif
Author/Authors :
Platts، نويسنده , , Michelle Y. and Barber، نويسنده , , Christopher G. and Chiva، نويسنده , , Jean-Yves and Eastwood، نويسنده , , Rachel L. and Fenwick، نويسنده , , David R. and Paradowski، نويسنده , , Kerry A. and Blakemore، نويسنده , , David C.، نويسنده ,
Issue Information :
هفته نامه با شماره پیاپی سال 2011
Pages :
3
From page :
512
To page :
514
Abstract :
An efficient route to dipyridone acid HIV integrase inhibitors is developed. The key steps include a one-pot three-step formation of the core template (containing one point of structural diversity) followed by a regioselective benzylation and in situ deprotection to afford the title compounds.
Keywords :
Dipyridone acid , integrase , Heterocycles , Antiviral agents , Ring-closure
Journal title :
Tetrahedron Letters
Serial Year :
2011
Journal title :
Tetrahedron Letters
Record number :
1876605
Link To Document :
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