Author/Authors :
Gan، نويسنده , , Haifeng and Lu، نويسنده , , Yunyu and Huang، نويسنده , , Yue and Ni، نويسنده , , Lijun and Xu، نويسنده , , Jinyi and Yao، نويسنده , , Hequan and Wu، نويسنده , , Xiaoming، نويسنده ,
Abstract :
An environmental-benign methodology to synthesize 1-benzoylisoquinolines from 1-benzyl-3, 4-dihydroisoquinolines or 1-benzyl-1,2,3,4-tetrahydroisoquinolines using dioxygen as an oxidant was developed. This methodology in combination with Bischler-Napieralski reaction leads to a facile synthesis of 1-benzoylisoquinolines from phenylacetic acids and phenylethanamines.