Author/Authors :
Kiyoi، نويسنده , , Yasuko and Laats، نويسنده , , Steven and Kiyoi، نويسنده , , Takao and Wishart، نويسنده , , Grant E. Brown، نويسنده , , Angus and Ray، نويسنده , , Peter، نويسنده ,
Abstract :
Hexahydro[2]benzopyrano[4,3-c]pyridines were synthesized by an intramolecular hetero Diels–Alder reaction. The reaction was applicable to a range of substrates and the products could be easily converted into serotonin 5-HT2C receptor agonists.
Keywords :
intramolecular hetero Diels–Alder reaction , 3-c]pyridines , Serotonin 5-HT2C receptor agonists , Microwave-assisted synthesis