• Title of article

    Stereoselective synthesis of tetrahydro-2H-[2]benzopyrano[3,4-c]pyrrol-3-ones and related compounds as precursors of serotonin 5-HT2C receptor agonists

  • Author/Authors

    Francis، نويسنده , , Stuart and Kiyoi، نويسنده , , Takao and Reid، نويسنده , , Mark and Davies، نويسنده , , Keneth and Laats، نويسنده , , Steven and McArthur، نويسنده , , Duncan and Feilden، نويسنده , , Helen and Easson، نويسنده , , Anna-Marie and Kiyoi، نويسنده , , Yasuko and Wishart، نويسنده , , Grant and Ray، نويسنده , , Peter، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2011
  • Pages
    5
  • From page
    3421
  • To page
    3425
  • Abstract
    Tetrahydro-2H-[2]benzopyrano[3,4-c]pyrrol-3-ones and the related 3a-methyl-2,3,3a,4,5,9b-hexahydro-1H-benzo[e]isoindole analogues were synthesised by an intramolecular Diels–Alder reaction. The observed stereoselectivity was dependent upon the nature of the tethered dienophile as well as the judicious placement of the amide.
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2011
  • Journal title
    Tetrahedron Letters
  • Record number

    1878640