Title of article
Palladium(II)-catalyzed oxidative Heck coupling of thiazole-4-carboxylates
Author/Authors
Li، نويسنده , , Ziyuan and Ma، نويسنده , , Ling and Tang، نويسنده , , Changhua and Xu، نويسنده , , Jinyi and Wu، نويسنده , , Xiaoming and Yao، نويسنده , , Hequan، نويسنده ,
Issue Information
هفته نامه با شماره پیاپی سال 2011
Pages
5
From page
5643
To page
5647
Abstract
Oxidative Heck coupling of thiazole-4-carboxylates via palladium(II)-catalyzed C–H bond activation has been achieved in moderate to good yields. No ligand, and no acidic additive were used in the reaction. The results showed that this protocol tolerated a series of substitutions on the thiazole ring. A preliminary attempt of direct arylation with p-xylene via Pd(II)-catalyzed C–H bond activation has also been done.
Keywords
C–H bond activation , Thiazole-4-carboxylate , Oxidative Heck-coupling , Direct arylation , Alkenylation
Journal title
Tetrahedron Letters
Serial Year
2011
Journal title
Tetrahedron Letters
Record number
1879433
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