Author/Authors :
Sun، نويسنده , , Jun and Zhang، نويسنده , , Xuefeng and Li، نويسنده , , Fulong and Ding، نويسنده , , Chunyong and Wu، نويسنده , , Wenjuan and Zhang، نويسنده , , Ao، نويسنده ,
Abstract :
Reaction of methyl 4,6-O-benzylidene-3(2)-deoxy-hexopyranosid-2(3)-ulose (1) with various arylamines under Bargellini reaction conditions was investigated. A series of unique enaminoketones 3–12 was obtained unexpectedly under basic conditions in 52–72% yield.
Keywords :
glycal , Arylamine , Bargellini reaction , base , Aminoglycosidation