• Title of article

    Regioselective ortho-acetoxylation/methoxylation of N-(2-benzoylphenyl)benzamides via substrate directed C–H activation

  • Author/Authors

    Reddy، نويسنده , , B.V. Subba and Revathi، نويسنده , , G. and Reddy، نويسنده , , A. Srinivas and Yadav، نويسنده , , J.S.، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2011
  • Pages
    4
  • From page
    5926
  • To page
    5929
  • Abstract
    A highly regioselective ortho-acetoxylation of N-(2-benzoylphenyl)benzamides has been achieved using a catalytic amount of Pd(OAc)2 (10 mol %) and a stoichiometric amount of PhI(OAc)2 in a mixture of acetic anhydride and acetic acid via C–H activation to produce the corresponding 2-acetoxybenzamides in good yields. ortho-Methoxylation has been accomplished using methanol under similar conditions.
  • Keywords
    ortho-Acetoxylation/methoxylation , Aromatic C–H activation , hypervalent iodine , Benzamide , Pd(II) catalysis
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2011
  • Journal title
    Tetrahedron Letters
  • Record number

    1879501