Title of article
Diastereoselective arylation of enantiopure 3-bromopiperidin-2-one derived from (R)-(−)-2-phenylglycinol with organocuprate reagents
Author/Authors
Romero، نويسنده , , Oscar and Castro، نويسنده , , Alejandro and Terلn، نويسنده , , Joel L. and Gnecco، نويسنده , , Dino and Orea، نويسنده , , Marيa L. and Mendoza، نويسنده , , ءngel and Flores، نويسنده , , Marcos and Roa، نويسنده , , Luis F. and Juلrez، نويسنده , , Jorge R.، نويسنده ,
Issue Information
هفته نامه با شماره پیاپی سال 2011
Pages
4
From page
5947
To page
5950
Abstract
The diastereoselective substitution of 3-bromolactam derived from (R)-(−)-2-phenylglycinol with a variety of arylcuprate reagents is presented. The stereochemical outcome of the substitution reaction is discussed. The method provides an efficient and straightforward route to enantiopure 3-arylpiperidines.
Journal title
Tetrahedron Letters
Serial Year
2011
Journal title
Tetrahedron Letters
Record number
1879506
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