• Title of article

    Effect of halogenation reagents on halocyclization and Overman rearrangement of allylic trichloroacetimidates

  • Author/Authors

    Liu، نويسنده , , Na and Schienebeck، نويسنده , , Casi M. and Collier، نويسنده , , Michelle D. and Tang، نويسنده , , Weiping، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2011
  • Pages
    3
  • From page
    6217
  • To page
    6219
  • Abstract
    Electrophilic halogen can promote either halocyclization or Overman rearrangement of allylic trichloroacetimidates. We found that the chemoselectivity was dependent on the nature of the halogenation reagents for primary allylic trichloroacetimidates. A one-pot procedure was developed for the preparation of allylic trichloroacetamides directly from allylic alcohols at room temperature.
  • Keywords
    Overman rearrangement , Allylic alcohols , Halocyclization , Allylic amide , Halogen
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2011
  • Journal title
    Tetrahedron Letters
  • Record number

    1879572