• Title of article

    Yb(OTf)3-promoted effective benzylation and allylation with N-tosyl amino group as a stable leaving group

  • Author/Authors

    Liu، نويسنده , , Jinqian and Wang، نويسنده , , Limin and Zheng، نويسنده , , Xingzhou and Wang، نويسنده , , Aili and Zhu، نويسنده , , Mengyun and Yu، نويسنده , , Jianjun and Shen، نويسنده , , Qiang، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2012
  • Pages
    4
  • From page
    1843
  • To page
    1846
  • Abstract
    A simple, inexpensive, environmentally friendly, and highly efficient benzylation and allylation of 1,3-dicarbonyl compounds with sulfonamides in the presence of Yb(OTf)3 is described. Yb(OTf)3 was proved to be a good catalyst for the cleavage of sp3 carbon–nitrogen bond. Various 1,3-dicarbonyl compounds can couple with a broad range of tosyl-activated benzylic and allylic amines to give diversely functionalized products in good to excellent yields.
  • Keywords
    3-Dicarbonyl compounds , N-tosyl amino group , Benzylation and allylation , Alkylation , Yb(OTf)3 , 1
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2012
  • Journal title
    Tetrahedron Letters
  • Record number

    1880442