• Title of article

    Solvent free, N,N′-carbonyldiimidazole (CDI) mediated amidation

  • Author/Authors

    Verma، نويسنده , , Sanjeev K. and Ghorpade، نويسنده , , Ramarao and Pratap، نويسنده , , Ajay and Kaushik، نويسنده , , M.P.، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2012
  • Pages
    4
  • From page
    2373
  • To page
    2376
  • Abstract
    The method involves CDI mediated amidation under solvent-free conditions. The protocol is green, simple, and scalable and has broad structural applicability. The protocol has also been used for BOC protection of amine. The protocol has reduced the time for CDI mediated amidation from 2–4 h to 5–10 min without the use of any dry organic solvent and nitrogen atmosphere.
  • Keywords
    Boc protection , green chemistry , CDI , Amidation
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2012
  • Journal title
    Tetrahedron Letters
  • Record number

    1880661