Title of article
Toward versatile methods leading to highly functionalized imidazo[1,2-a]pyridines
Author/Authors
Basilio-Lopes، نويسنده , , Alexandra and de Aquino، نويسنده , , Thiago Mendonça and Mongeot، نويسنده , , Alexandre and Bourguignon، نويسنده , , Jean-Jacques and Schmitt، نويسنده , , Martine، نويسنده ,
Issue Information
هفته نامه با شماره پیاپی سال 2012
Pages
5
From page
2583
To page
2587
Abstract
A convenient and general method of preparation of polyfunctionalized imidazo[1,2-a]pyridines is reported. This methodology involves activation of secondary amides leading to the formation of the corresponding amidines 9. Different activating reagents have been evaluated and the efficiency of PCl5 was illustrated with alkyl functionalized groups.
Keywords
PCl5 , 2-a]pyridine , Amidines , TiCl4
Journal title
Tetrahedron Letters
Serial Year
2012
Journal title
Tetrahedron Letters
Record number
1880752
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