• Title of article

    Tetrahydroquinazoline-substituted chromones from Diels–Alder reaction of (E)-2-styrylchromones and pyrimidine ortho-quinodimethane

  • Author/Authors

    Patoilo، نويسنده , , Diana T. and Silva، نويسنده , , Artur M.S. and Pinto، نويسنده , , Diana C.G.A. and Santos، نويسنده , , Clementina M.M. and Tomé، نويسنده , , Augusto C. and Cavaleiro، نويسنده , , José A.S.، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2012
  • Pages
    4
  • From page
    2722
  • To page
    2725
  • Abstract
    The Diels–Alder reaction of (E)-2-styrylchromones with a pyrimidine ortho-quinodimethane is reported for the first time. These cycloaddition reactions afford mixtures of two regioisomeric tetrahydroquinazoline-substituted chromones in moderate to excellent global yields. Irrespective of the substituents on the 2-styrylchromones, the 2-(7-aryl-4-methoxy-2-methyl-5,6,7,8-tetrahydroquinazolin-6-yl)chromone derivatives are always the major isomers.
  • Keywords
    Tetrahydroquinazolines , Cycloadditions , 2-Styrylchromones , Pyrimidine ortho-quinodimethane , NMR
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2012
  • Journal title
    Tetrahedron Letters
  • Record number

    1880814