• Title of article

    Regioselective assembly of 3,4-dihydroisoquinoline derivatives

  • Author/Authors

    Gao، نويسنده , , Zhongli and Davis، نويسنده , , Larry and Chiang، نويسنده , , Yulin and Munson، نويسنده , , Randall and Hendrix، نويسنده , , James A.، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2012
  • Pages
    4
  • From page
    4429
  • To page
    4432
  • Abstract
    A facile two-step sequence (9→10→1) of regioselective assembly of 3,4-dihydroisoquinoline derivatives 1 is reported. The halogen derivatives provide opportunity for Suzuki, Buchwald, and related coupling reactions useful for expanding the scaffold and lead optimization in drug discovery.
  • Keywords
    Alkaloids , Bischler–Napieralski reaction , Pictet–Spengler reaction , 3 , 4-Dihydroisoquinoline
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2012
  • Journal title
    Tetrahedron Letters
  • Record number

    1881557

    • Link To Document
    https://search.isc.ac/dl/search/defaultta.aspx?DTC=10&DC=1881557