• Title of article

    Ru(II)-Pheox catalyzed N–H insertion reaction of diazoacetamides: synthesis of N-substituted α-aminoamides

  • Author/Authors

    Soda Chanthamath، نويسنده , , Soda and Thongjareun، نويسنده , , Songkharm and Shibatomi، نويسنده , , Kazutaka and Iwasa، نويسنده , , Seiji، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2012
  • Pages
    4
  • From page
    4862
  • To page
    4865
  • Abstract
    An efficient protocol for the preparation of α-aminoamides was developed via the Ru(II)-dm-Pheox catalyzed N–H insertion reaction of various diazoacetamides with several amines, including aniline. This catalytic N–H insertion reaction was also applied to the synthesis of 2-(2-methylquinolin-4-ylamino)-N-phenylacetamide, a potential antileishmanial agent.
  • Keywords
    Ruthenium catalyst , ?-Aminoamide , N–H insertion reaction , Diazoacetamide
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2012
  • Journal title
    Tetrahedron Letters
  • Record number

    1881728