• Title of article

    Organocatalytic synthesis of novel purine and pyrimidine acyclic nucleosides

  • Author/Authors

    Palazzolo، نويسنده , , Martيn A. and Pérez-Sلnchez، نويسنده , , Marيa and Iribarren، نويسنده , , Adolfo M. and Lewkowicz، نويسنده , , Elizabeth S. and Domيnguez de Marيa، نويسنده , , Pablo، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2012
  • Pages
    4
  • From page
    6797
  • To page
    6800
  • Abstract
    Organocatalysis is assessed for the first time in the synthesis of purine and pyrimidine acyclic nucleosides providing high yields and straightforward work-up procedures. Nucleobases containing aldehydes are catalytically ligated (C–C bond formation) to acetone or to phosphonate-containing ketones by means of pyrrolidine or silica-immobilized piperazine as amine-based organocatalysts.
  • Keywords
    Piperazine , acyclic nucleosides , organocatalysis , pyrrolidine , Phosphonate
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2012
  • Journal title
    Tetrahedron Letters
  • Record number

    1882950