Author/Authors :
Davey، نويسنده , , Paul R.J. and Delouvrié، نويسنده , , Bénédicte and Dorison-Duval، نويسنده , , Delphine and Germain، نويسنده , , Hervé and Harris، نويسنده , , Craig S. and Magnien، نويسنده , , Françoise and Ouvry، نويسنده , , Gilles and Tricotet، نويسنده , , Thomas، نويسنده ,
Abstract :
The preparation of N-2 substituted 2H-1,2,3-triazoles substituted at C-4 with an organometallic moiety has no recognised precedent. Herein, we report their efficient preparation via CH borylation and demonstrate their successful application to aryl–aryl Suzuki cross-coupling.
Keywords :
2 , 3-Triazole 4-boronates , Direct CH borylation , Suzuki–Miyaura cross-coupling , 2H-1