• Title of article

    A practical one-pot procedure for the synthesis of N–H isoquinolones

  • Author/Authors

    Lu، نويسنده , , Shaonan and Lin، نويسنده , , Yingfu and Zhong، نويسنده , , Hongban and Zhao، نويسنده , , Kang and Huang، نويسنده , , Jianhui، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2013
  • Pages
    5
  • From page
    2001
  • To page
    2005
  • Abstract
    A practical one-pot procedure for the preparation of N–H isoquinolones has been developed. This 2-step process via C–H activation of N-alkoxyl benzamides and NaH-mediated dealkoxylation reaction has been demonstrated to be a high yielding alternative methodology for the efficient synthesis of a wide range of representative N–H isoquiolones. In addition, the experimental precedent supported mechanism of the dealkoxylation reaction was also proposed.
  • Keywords
    Isoquinolone , C–H activation , Organometallics , Pd-catalysis , N–O bond cleavage
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2013
  • Journal title
    Tetrahedron Letters
  • Record number

    1884193