• Title of article

    Convenient one-pot synthesis of N3-substituted pyrido[2,3-d]-, pyrido[3,4-d]-, pyrido[4,3-d]-pyrimidin-4(3H)-ones, and quinazolin-4(3H)-ones analogs

  • Author/Authors

    Deau، نويسنده , , Emmanuel and Hédou، نويسنده , , Damien and Chosson، نويسنده , , Elizabeth and Levacher، نويسنده , , Vincent and Besson، نويسنده , , Thierry، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2013
  • Pages
    4
  • From page
    3518
  • To page
    3521
  • Abstract
    A convenient microwave-assisted one-pot sequential synthesis provided access to novel pyridopyrimidin-4-(3H)-ones in good to excellent yields. Anthranilic acid, 2- and 4-aminonicotinic acids, and 3-aminoisonicotinic acid were quantitatively converted into the analogous amidinoesters which undergo rapid cyclization in the presence of an amine.
  • Keywords
    microwave-assisted chemistry , 3-d]-pyrimidin-4(3H)-ones , 4-d]-pyrimidin-4(3H)-ones , 3-d]-pyrimidin-4(3H)-ones , One-pot sequential synthesis
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2013
  • Journal title
    Tetrahedron Letters
  • Record number

    1884833