Title of article :
A convenient method for the one-step synthesis of phosphonic peptides
Author/Authors :
Skore?ski، نويسنده , , Marcin and Oleksyszyn، نويسنده , , J?zef and Sie?czyk، نويسنده , , Marcin، نويسنده ,
Issue Information :
هفته نامه با شماره پیاپی سال 2013
Abstract :
A novel and efficient method for the synthesis of peptidyl derivatives of 1-aminoalkylphosphonate diaryl esters is presented. Phosphonic peptides were obtained in one step via an amidoalkylation reaction using amides of N-protected amino acids or peptides, triphenyl phosphite, and an appropriate aldehyde.
Keywords :
1-Aminoalkylphosphonates , Phosphonic peptides , Amides , Amidoalkylation , serine protease inhibitors
Journal title :
Tetrahedron Letters
Journal title :
Tetrahedron Letters
