• Title of article

    RGD-conjugated triarylmethyl radical as probe for electron paramagnetic imaging

  • Author/Authors

    Patrice Driesschaert، نويسنده , , Benoît and Levêque، نويسنده , , Philippe and Gallez، نويسنده , , Bernard and Marchand-Brynaert، نويسنده , , Jacqueline، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2013
  • Pages
    3
  • From page
    5924
  • To page
    5926
  • Abstract
    A stable RGD-conjugated triarylmethyl (TAM) radical 3 has been synthesized in a straightforward three-step sequence. CT-03 ‘the Finland trityl’ which is a very popular contrast agent for electron paramagnetic resonance imaging has been covalently bound to the NH2-ending of a pentapeptide commonly used to target integrins and confers tissue selectivity. Moreover, this new TAM radical is stable and sensitive to molecular oxygen.
  • Keywords
    EPR , Trityl radical , RGD , Oximetry
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2013
  • Journal title
    Tetrahedron Letters
  • Record number

    1886423