• Title of article

    Synthesis of novel 5-oxaprotoberberines as bioisosteres of protoberberines

  • Author/Authors

    Jin، نويسنده , , Yifeng and Khadka، نويسنده , , Daulat Bikram and Yang، نويسنده , , Su Hui and Zhao، نويسنده , , Chao and Cho، نويسنده , , Won-Jea Cho، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2014
  • Pages
    4
  • From page
    1366
  • To page
    1369
  • Abstract
    5-Oxaprotoberberinones and 5-oxaprotoberberinium were synthesized as bioisosteres of protoberberines. 5-Oxaprotoberberinones were prepared by linking phenol with the isoquinolone ring of 3-phenolisoquinolones by methyleneoxy bridge, while the quaternary 5-oxaprotoberberinium salt was synthesized by reduction and oxidation of the lactam moiety of 5-oxaprotoberberinone.
  • Keywords
    Bioisostere , 5-Oxaprotoberberinium , Protoberberine , 5-Oxaprotberberin-8-one
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2014
  • Journal title
    Tetrahedron Letters
  • Record number

    1888233